Antithrombotics

Effects

  • Antithrombotic
  • Anticoagulant
  • Fibrinolytic

Active ingredients

Salicylates:

P2Y12 antagonists:

GP IIb/IIIa antagonists:

  • Abciximab (ReoPro)
  • Eptifibatide (Integrilin)
  • Tirofiban (Aggrastat)

PAR-1 antagonists:

  • Vorapaxar (Zontivity)

Vitamin K antagonists (coumarins):

  • Phenprocoumon (Marcoumar).
  • Acenocoumarol (Sintrom)
  • Not on sale in many countries: dicoumarol, warfarin.

Heparins:

  • Heparin sodium
  • Heparin-Calcium (Calciparine)
  • Certoparin (Sandoparin)
  • Dalteparin (Fragmin)
  • Enoxaparin (Clexane)
  • Nadroparin (Fraxiparine, Fraxiforte)

Fibrinolytics:

  • Alteplase
  • Urokinase
  • Streptokinase

Thrombin inhibitors:

  • Leech: hirudin
  • Bivalirudin (Angiox)
  • Lepirudin (Refludan, out of commerce).
  • Argatroban (Argatra)
  • Dabigatran (Pradaxa)

Factor Xa inhibitors:

  • Rivaroxaban (Xarelto)
  • Apixaban (Eliquis)
  • Edoxaban (Savaysa)

DOAK:

  • Factor Xa inhibitors
  • Thrombin inhibitors

Other: