Bambuterol

Products

Bambuterol is commercially available in the form of tablets (Bambec). The drug is not registered in many countries.

Structure and properties

Bambuterol (C18H29N3O5, Mr = 367.4 g/mol) is present in drugs as bambuterol hydrochloride. It is a prodrug of terbutaline.

Effects

Bambuterol (ATC R03CC12) is bronchodilator. Its effects are due to stimulation of adrenergic β2-receptors in bronchial muscles. The active metabolite is terbutaline.

Indications

Prevention and treatment of respiratory diseases associated with airway constriction due to bronchial muscle spasm (obstructive airway disease).