Effects Nifedipine is an active ingredient of the dihydropyridine group and has a relaxing effect on vascular smooth muscle. When used topically or orally, it dilates blood vessels, improves blood flow and thus wound healing, is anti-inflammatory, and relieves anal sphincter spasms. Dihydropyridines inhibit the influx of calcium into smooth muscle cells by inhibiting L-type … Nifedipine Cream for Anal Fissure
Symptoms Anal fissure is a tear or cut in the skin of the anal canal. This results in severe pain that occurs during and up to several hours after defecation. It may radiate locally and be accompanied by an uncomfortable itching sensation. Fresh blood can often be seen on toilet paper or stool. Causes Possible … Anal Fissure: Symptoms, Diagnosis, Causes and Treatment
Products Remifentanil is commercially available as a powder for the preparation of a concentrate for solution for injection or infusion (Ultiva, generic). It has been approved in many countries since 1996. Structure and properties Remifentanil (C20H28N2O5, Mr = 376.4 g/mol) is present in drugs as remifentanil hydrochloride, a white powder. The drug is rapidly hydrolyzed … Remifentanil
Products Cinnarizine and dimenhydrinate are commercially available as a fixed combination in the form of tablets (Arlevert). The drug has been on the market in many countries since 2012. It was available earlier in Germany. Structure and properties The drug consists of 3 molecules in total. Dimenhydrinate is a combination of diphenhydramine and chlorotheophyllin. Effects … Cinnarizine and Dimenhydrinate
General information Amlodipine is an antihypertensive drug. In addition to its use as a basic medication for high blood pressure (arterial hypertension), it is also used to treat chronic tightness in the chest (angina pectoris) and to prevent acute attacks of angina pectoris in Prinzmetal angina. Pharmacologically, it belongs to the class of calcium channel … Amlodipine
What should I watch out for when stopping this medicine? Amlodipine is one of the drugs that lower blood pressure. All drugs in this group must not be suddenly discontinued. Taking the drug reduces the number of so-called receptors in the body, which otherwise keep blood pressure low. The body needs some time to readjust … What should I watch out for when stopping this medicine? | Amlodipine
Contraindications Amlodipine should only be given with special caution to patients with a narrowing of the aortic valve (see aortic valve stenosis), as the drug’s blood pressure-lowering effect can lead to reduced blood flow to the heart, which in turn could trigger a heart attack. In patients with a damaged liver, a lower starting dose … Contraindications | Amlodipine
Are amlodipine tablets halvable? The divisibility of amlodipine tablets depends on the preparation. In the package insert it is noted in each case if the tablets can be divided in half. For example, the tablets of the preparation Amlodipine – 1 A Pharma® 5mg Tablets N can be divided in half. Amlodipine tablets are available … Are amlodipine tablets halvable? | Amlodipine
Products Imepitoin is commercially available in tablet form (Pexion). It has been approved in many countries since 2013. Structure and properties Imepitoin (C13H14ClN3O2, Mr = 279.7 g/mol) is a morpholine and imidazolone derivative. It is structurally unrelated to the benzodiazepines. Effects Imepitoin (ATCvet QN03AX90) has antiepileptic properties. Its effects are due to partial agonism with … Imepitoin
Synonyms in a broader sense Calcium channel blocker English: antagonist of calcium Definition Calcium antagonists have an opposite effect to calcium: they prevent calcium from reaching the cells of the heart muscle, the cells of the electrical conduction system (the heart’s electrical conduction system) at the heart and the muscle cells of the blood vessels. … Calcium antagonists
What are the alternatives to calcium antagonists? The answer to the question what the alternatives to calcium antagonists are depends mainly on the purpose for which the drug is to be taken. In the treatment of high blood pressure, for example, there are several alternatives that can be chosen. In addition to the so-called ACE … What are the alternatives to calcium antagonists? | Calcium antagonists
Calcium antagonists in Parkinson’s disease Calcium antagonists should not be used in people with Parkinson’s disease. Research has shown that certain members of this group of drugs can worsen the symptoms typical of the disease. However, there are also studies that suggest that a particular calcium channel blocker may have a positive effect on the … Calcium antagonists in Parkinson’s disease | Calcium antagonists
