Tramadol – what the active ingredient can do

How tramadol works Tramadol is a pain-relieving (analgesic) substance from the opioid group. Humans have an endogenous analgesic system that is activated in stressful situations, among other things. For example, after serious accidents, injured people are often initially able to help others without even noticing their own injury. In addition, the analgesic prevents the reuptake … Tramadol – what the active ingredient can do

Cyclobenzaprine

Products Cyclobenzaprine is commercially available in the United States and elsewhere in the form of film-coated tablets. No finished drug products containing cyclobenzaprine are currently registered in many countries. Structure and properties Cyclobenzaprine (C20H21N, Mr = 275.4 g/mol) is present in drugs as cyclobenzaprine hydrochloride, a white crystalline powder that is soluble in water. It … Cyclobenzaprine

Tramadol Combats Severe Pain

Tramadol is an analgesic used to fight moderate and severe pain. However, the active ingredient only combats the symptoms, not the cause of the pain. Tramadol comes in the form of tablets, drops, and suppositories, as well as injections and infusions. Just like other painkillers, tramadol has side effects: It should be especially noted – … Tramadol Combats Severe Pain

Tramadol: Drug Effects, Side Effects, Dosage and Uses

Products Tramadol is commercially available in the form of tablets, capsules, melting tablets, drops, effervescent tablets, suppositories, and as a solution for injection. (Tramal, generic). Fixed combinations with acetaminophen are also available (Zaldiar, generic). Tramadol was developed by Grünenthal in Germany in 1962 and has been approved in many countries since 1977 and in the … Tramadol: Drug Effects, Side Effects, Dosage and Uses

Tramadol and Paracetamol

Products The combination drug containing the active ingredients tramadol and paracetamol is commercially available in the form of film-coated tablets (Zaldiar). It has been approved in many countries since 2002. In 2014, generic versions went on sale. The effervescent tablets are out of trade. Structure and properties Tramadol (C16H25NO2, Mr = 263.38 g/mol) is a … Tramadol and Paracetamol

Enantiomers

Introductory question How much active ingredient is in a 10 mg cetirizine tablet? (a) 5 mg B) 7.5 mg C) 10 mg The correct answer is a. Image and mirror image Many active pharmaceutical ingredients exist as racemates. They consist of two molecules that behave like an image and mirror image of each other. These … Enantiomers

Ondansetron

Products Ondansetron is commercially available in the form of film-coated tablets, meltable tablets (lingual tablets), as a syrup, and as an infusion/injection preparation. In addition to the original Zofran, generic versions are also available. Ondansetron was introduced in 1991 as the first active ingredient from the group of 5-HT3 receptor antagonists was approved. Structure and … Ondansetron

Paracetamol: Drug Effects, Side Effects, Dosage and Uses

Products Paracetamol is commercially available in the form of tablets, film-coated tablets, melting tablets, effervescent tablets, as granules, drops, syrups, suppositories, soft capsules, and infusion solution, among others (e.g., Acetalgin, Dafalgan, Panadol, and Tylenol). Paracetamol was not approved until the 1950s (Panadol, Tylenol), although it was developed in the 19th century. It has been registered … Paracetamol: Drug Effects, Side Effects, Dosage and Uses

Knee Osteoarthritis

Symptoms Knee osteoarthritis manifests itself as knee pain, which occurs primarily during physical activity and when the joint is under stress. They are often triggered at the beginning of movement (start-up pain), when climbing stairs, when standing up or when walking longer distances. Other complaints include limitation of mobility and quality of life, instability, an … Knee Osteoarthritis

Fibromyalgia Causes and Treatment

Symptoms Fibromyalgia is a chronic, noninflammatory disorder that manifests as pain throughout the body and is characterized by numerous other complaints. It is much more common in women than in men and usually first appears in middle age. Chronic, bilateral, diffuse pain. Muscle pain, pain in the limbs, back pain, joint pain, neck pain, headaches, … Fibromyalgia Causes and Treatment

Venlafaxine: Drug Effects, Side Effects, Dosage and Uses

Products Venlafaxine is commercially available in tablet and sustained-release capsule form. In addition to the original Efexor ER (USA: Effexor XR), generic versions are also available. The active ingredient was approved in many countries in 1997. Structure and properties Venlafaxine (C17H27NO2, Mr= 277.4 g/mol) is a bicyclic phenylethylamine and cyclohexanol derivative that is structurally closely … Venlafaxine: Drug Effects, Side Effects, Dosage and Uses