Parasympatholytics

Products Parasympatholytics are commercially available, for example, in the form of tablets, capsules, solutions, as inhalation preparations, injection solutions, and eye drops. This article refers to antagonists at muscarinic acetylcholine receptors. Antagonists at nicotinic acetylcholine receptors, such as ganglion blockers, are discussed separately. Structure and properties Many parasympatholytics are structurally derived from atropine, a natural … Parasympatholytics

Spasmolytics

Products Spasmolytics are commercially available in the form of tablets, suppositories, and injectables, among others. In many countries, scopolamine butylbromide is among the best-known representatives. Structure and properties Spasmolytics are often derived from the tropane alkaloids atropine and scopolamine from nightshade plants or from the benzylisoquinoline papaverine from the opium poppy. Effects Spasmolytics have spasmolytic … Spasmolytics

Drofenin

Products Drofenine is registered for export in tablet form (Lunadon, combination). It has been approved in many countries since 1977 but is not commercially available. Structure and properties Drofenine (C20H31NO2, Mr = 317.47 g/mol) is a derivative of atropine. It exists as drofenine hydrochloride, a white, loose crystalline powder that is very soluble in water. … Drofenin