Diphenoxylate

Products Diphenoxylate is not commercially available in many countries. Combination products with atropine sulfate are commercially available in the United States. Structure and properties Diphenoxylate (C30H32N2O2, Mr = 452.6 g/mol) is present in drugs as diphenoxylate hydrochloride, a white crystalline powder that is very sparingly soluble in water. It is a derivative of pethidine and … Diphenoxylate

Difenoxin

Products Difenoxin is not commercially available in many countries. Structure and properties Difenoxin (C28H28N2O2, Mr = 424.5 g/mol) is the active metabolite of diphenoxylate and structurally related to loperamide (Imodium). Effects Difenoxin (ATC A07DA04) is peristaltic inhibitory and antidiarrheal. Indication Diarrhea