Sugammadex

Products

Sugammadex is commercially available as a solution for injection (Bridion). It was approved in many countries in January 2010.

Structure and properties

Modified gamma-cyclodextrin.

Effects

Sugammadex (ATC V03AB35) forms a complex with the neuromuscular blocking agents rocuronium or vecuronium in plasma, thus abolishing their effects.

Indications

Abrogation of neuromuscular blockade induced by rocuronium or vecuronium.