Valproate: Effects, Uses & Risks

Valproate is widely used in medicine to prevent seizures in epilepsy. In addition, it is often used as a phase prophylactic in bipolar disorder and schizoaffective psychosis. What is valproate? Valproate is widely used in medicine to prevent seizures in epilepsy. Valproates are salts of artificially produced valproic acid, which chemically belongs to the branched … Valproate: Effects, Uses & Risks

Tipranavir: Effects, Uses & Risks

The active medical ingredient Tipranavir is a drug that is used to treat people with HIV type 1. It is used as part of a combination antiretroviral therapy. The drug Tipranavir is available on the pharmacological market under the trade name Aptivus and is distributed by the producer Boehringer. The active ingredient tipranavir is considered … Tipranavir: Effects, Uses & Risks

Bromazepam

Products Bromazepam is commercially available in tablet form (Lexotanil). It has been approved in many countries since 1974. Structure and properties Bromazepam (C14H10BrN3O, Mr = 316.2 g/mol) exists as a white to yellowish crystalline powder that is practically insoluble in water. It is a brominated 1,4-benzodiazepine. Effects Bromazepam (ATC N05BA08) has antianxiety, sedative, and depressant … Bromazepam

Clonazepam

Products Clonazepam is commercially available as tablets, injectable solution, and oral drops (Rivotril). It has been approved in many countries since 1973. In the United States, it is marketed as Klonopin. Structure and properties Clonazepam (C15H10ClN3O3, Mr = 315.7 g/mol) exists as a faint yellowish crystalline powder that is practically insoluble in water. It is … Clonazepam

Flunitrazepam

Products Flunitrazepam is commercially available in the form of film-coated tablets (Rohypnol). It has been approved in many countries since 1975. Structure and properties Flunitrazepam (C16H12FN3O3, Mr = 313.3 g/mol) is a lipophilic, fluorinated and nitrated 1,4-benzodiazepine. It exists as a white to yellowish crystalline powder that is practically insoluble in water. Effects Flunitrazepam (ATC … Flunitrazepam

Rebound Effect: Function, Tasks, Role & Diseases

The rebound effect is specifically important after discontinuation of a prolonged medication. Mechanisms originally intended for the body’s adaptation can lead to undesirable side effects in medicine and other fields. What is the rebound effect? The rebound effect is a consequence of giving up a habit. In medicine, the focus here is when a medication … Rebound Effect: Function, Tasks, Role & Diseases

Dyes in Medicines

Which dyes are used? Coloring agents that are also used as food additives (E-numbers) are usually used for medicines. Which colorants are permitted depends on the legislation of the relevant countries. For Switzerland, the specifications published in the Medicines Approval Ordinance (AMZV), in Pharmacopoea Helvetica and in the Additives Ordinance apply. The following list shows … Dyes in Medicines

Lorazepam: Effects, Uses & Risks

Lorazepam is a substance in the benzodiazepine group. It is used as an anxiolytic, sedative, hypnotic, anticonvulsant, and muscle relaxant. Furthermore, lorazepam is misused in the drug scene. It is subject to narcotics laws when the amount of active ingredient exceeds 2.5 mg per unit. What is lorazepam? Lorazepam is a drug present as a … Lorazepam: Effects, Uses & Risks

Lopinavir: Effects, Uses & Risks

Lopinavir is a drug used in the therapy of HIV infection, acting as a protease inhibitor. The HIV protease inhibitor is used in combination with AbbVie’s product ritonavir and is known on the market by the trade name Kaletra. The drug received approval from the relevant EU Commission in 2001. What is lopinavir? Lopinavir is … Lopinavir: Effects, Uses & Risks

Diazepam Nasal Spray

Products Valtoco diazepam nasal spray was approved in the United States in 2020. The benzodiazepine diazepam has been available in other dosage forms since the 1960s. Structure and properties Diazepam (C16H13ClN2O, Mr = 284.7 g/mol) is a lipophilic benzodiazepine. It exists as a white crystalline powder that is very sparingly soluble in water. Effects Diazepam … Diazepam Nasal Spray

Chlordiazepoxide

Products Chlordiazepoxide was synthesized in the 1950s by Leo Sternbach at Hoffmann-La Roche and became the first active ingredient in the benzodiazepine group to be marketed in 1960 (Librium). In many countries, it is currently only available in combination with clidinium bromide or amitriptyline (Librax, Limbitrol). In other countries, the monopreparation Librium is still available. … Chlordiazepoxide

Nelfinavir: Effects, Uses & Risks

The pharmacological substance nelfinavir is a drug that is counted among the so-called HIV protease inhibitors. It is available on the medical market under the trade name Viracept. The drug Nelfinavir is indicated for antiretroviral therapy of patients infected with HIV-1. The special protease inhibitors are used as part of a so-called ‘highly active antiretroviral … Nelfinavir: Effects, Uses & Risks