Ebastine: Effects, Side Effects

How does ebastine work? Ebastine has an anti-allergic effect by inhibiting the activation of histamine H1 receptors by histamine. In the course of allergic reactions, this messenger substance is released in large quantities. By docking at its binding sites, it triggers allergic symptoms such as sneezing and itching. By occupying the histamine binding sites, ebastine … Ebastine: Effects, Side Effects

Antihistamines for Allergies

Products Antihistamines are often taken in the form of tablets. In addition, drops, solutions, lozenges, capsules, gels, creams, eye drops, nasal sprays, and injectable solutions are also available, among others. The first active ingredient from this group was phenbenzamine (Antergan), developed in France in the 1940s. It is no longer commercially available today. Structure and … Antihistamines for Allergies

Ebastine

Products Ebastine is commercially available in the form of film-coated tablets (e.g., Ebastel). The drug is not registered in many countries. Structure and properties Ebastine (C32H39NO2, Mr = 469.7 g/mol) Effects Ebastine (ATC R06AX22) has antiallergic properties. It is not anticholinergic and barely crosses the blood–brain barrier. Indications For symptomatic treatment of seasonal and perennial … Ebastine