Beta Blocker Effects and Side Effects

Products Beta-blockers are available in many countries in the form of tablets, film-coated tablets, sustained-release tablets, as capsules, solution, eye drops, and as injection and infusion solutions. Propranolol (Inderal) was the first representative of this group to appear on the market in the mid-1960s. Today, the most important active ingredients include atenolol, bisoprolol, metoprolol and … Beta Blocker Effects and Side Effects

Celiprolol

Products Celiprolol is commercially available in the form of film-coated tablets (Selectol). It has been approved in many countries since 1987. Structure and properties Celiprolol (C20H34ClN3O4, Mr = 415.95 g/mol is a racemate and is present in drugs as celiprolol hydrochloride, a white to pale yellow crystalline powder that is readily soluble in water. Effects … Celiprolol

P-Glycoprotein

P-glycoprotein P-glycoprotein (P-gp, MDR1) is a primary active efflux transporter with a molecular weight of 170 kDa, belonging to the ABC superfamily and consisting of 1280 amino acids. P-gp is the product of the -gene (formerly: ). P is for , ABC is for . Occurrence P-glycoprotein is found on various tissues of the human … P-Glycoprotein

Celiprolol: Effects, Uses & Risks

Celiprolol is a drug used to treat high blood pressure and coronary artery disease. The drug belongs to the beta-blocker group. It is predominantly used in combination with others rather than as a stand-alone medication. Celiprolol can cause various side effects or interactions. The use of the drug must always be in consultation with the … Celiprolol: Effects, Uses & Risks