Toremifene

Products

Toremifene is commercially available in tablet form (Fareston). It was approved in many countries in 1996 and went off the market in 2012.

Structure and properties

Toremifene (C26H28ClNO, 405.96 g/mol)

Effects

Toremifene (ATC L02BA02) is antiestrogenic.

Indications

Local unresectable, locally recurrent, or metastatic postmenopausal breast carcinoma (breast cancer).

Contraindications

For complete precautions, see the drug label.

Adverse effects

The most common adverse effects are hot flashes. Increased sweating, nausea, and leukorrhea are common.