narcotics

Propofol (Diprivan): Drug Effects, Side Effects, Dosage and Uses

Products Propofol is commercially available as an emulsion for injection or infusion (Disoprivan, generic). It has been approved in many countries since 1986. Structure and properties Propofol obtained by distillation (C12H18O, Mr = 178.3 g/mol, 2,6-diisopropylphenol) is a colorless to pale yellow, clear liquid that is sparingly soluble in water and miscible with hexane and … Propofol (Diprivan): Drug Effects, Side Effects, Dosage and Uses

Codeine: Drug Effects, Side Effects, Dosage and Uses

Products Codeine is available alone or in combination with other active ingredients in the form of tablets, effervescent tablets, capsules, dragées, syrups, drops, bronchial pastilles, and as suppositories. It is also combined fixedly with acetaminophen for the treatment of pain (see under codeine acetaminophen). Structure and properties Codeine (C18H21NO3, Mr = 299.36 g/mol) is -methylated … Codeine: Drug Effects, Side Effects, Dosage and Uses

Sedative

Products Sedatives are commercially available in the form of tablets, melting tablets, drops, as injectables and tinctures, among others. Structure and properties Sedatives do not have a uniform chemical structure. Effects The active ingredients have sedative properties. Some are additionally antianxiety, sleep-inducing, antipsychotic, antidepressant, and anticonvulsant. The effects are due to promotion of inhibitory mechanisms … Sedative

Narcotics Effects and Side Effects

Products The narcotics are a group of centrally acting drugs and substances, which are strongly regulated and controlled by the state respectively by the drug and health authorities. This is primarily to prevent abuse and to protect the population from the undesirable effects and addiction. Certain narcotics – for example, many potent hallucinogens – are … Narcotics Effects and Side Effects

Carfentanil

Products In many countries, no drugs containing carfentanil are on the market. The active ingredient is used in veterinary medicine (Wildnil). Legally, it belongs to narcotics. Structure and properties Carfentanil (C24H30N2O3, Mr = 394.5 g/mol) is structurally closely related to fentanyl, being 4-methoxycarbonylfentanyl. Carfentanil citrate is present in pharmaceuticals. The active ingredient was developed at … Carfentanil

Lisdexamphetamine

Products Lisdexamphetamine (LDX) was approved in many countries in March 2014 in capsule form (Elvanse). It has been available in the United States since 2007 (Vyvanse). The dosage form is non-retarded, unlike other ADHD medications. Continuous release is achieved with the conversion of the prodrug. Lisdexamphetamine is legally classified as a narcotic and therefore requires … Lisdexamphetamine

Embutramid

Products Embutramide is commercially available as a solution for injection as a combination preparation with the muscle relaxant mebezonium iodide and the local anesthetic tetracaine (T 61). It has been approved in many countries since 1971. Structure and properties Embutramide (C17H27NO3, Mr = 293.4 g/mol) is a derivative of γ-hydroxybutyric acid. Effects Embutramide (ATCvet QN51AX50) … Embutramid

Alfentanil

Products Alfentanil is commercially available as a solution for injection (Rapifen). It has been approved in many countries since 1983. Structure and properties Alfentanil (C21H32N6O3, Mr = 416.5 g/mol) is a 4-anilidopiperidine and a tetrazole derivative. It is present in the drug as alfentanil hydrochloride, a white powder that is readily soluble in water. The … Alfentanil

Dimenhydrinate

Products Dimenhydrinate is commercially available in the form of tablets, dragées, [chewing gum dragées>chewing gum], and capsules, among others. Since 2012, a combination with the calcium channel blocker cinnarizine has been approved in many countries (Arlevert) see under Cinnarizine and Dimenhydrinate. Structure and properties Dimenhydrinate (C24H28ClN5O3, Mr = 470.0 g/mol) is the salt of diphenhydramine … Dimenhydrinate

Aphrodisiacs

Effects Aphrodisiac Medical indications To promote sex drive or potency. Erectile dysfunction in men “Hypoactive Sexual Desire Disorder” (decreased sexual drive). Active ingredients Use v.a. in erectile dysfunction: phosphodiesterase-5 inhibitors increase blood flow to the corpus cavernosum of the penis and act only during sexual stimulation: Sildenafil (Viagra) Tadalafil (Cialis) Vardenafil (Levitra) Prostaglandins must be … Aphrodisiacs

Orexin Receptor Antagonists

Products Orexin receptor antagonists are commercially available in tablet form. The first agent in this group to be approved in the United States was suvorexant (Belsomra) in 2014. Lemborexant (Dayvigo) followed in 2019. Structure and properties Orexin receptor antagonists are characterized by a central ring structure to which heterocycles are attached on both sides. Effects … Orexin Receptor Antagonists