Products Meclozine is marketed as a fixed combination with caffeine and the vitamin pyridoxine in the form of capsules and suppositories (Itinerol B6). It has been approved in many countries since 1953. In some countries, the active ingredient is also called. Itinerol dragées went out of commerce in 2015. Structure and properties Meclozine (C25H27ClN2, Mr … Meclozin
Products Lorazepam is commercially available as tablets, meltable tablets, and a solution for injection. In addition to the original Temesta, generics and a combination product with the sedative antihistamine diphenhydramine are also available (Somnium). Lorazepam has been approved in many countries since 1973. Structure and properties Lorazepam (C15H10Cl2N2O2, Mr = 321.2 g/mol) is a white … Lorazepam
Products Lormetazepam is commercially available in tablet form (Loramet). Both drugs have been approved in many countries since 1981. Noctamide is no longer marketed. Structure and properties Lormetazepam (C16H12Cl2N2O2, Mr = 335.18 g/mol) is an -methylated lorazepam (Temesta). It belongs to the 5-aryl-1,4-benzodiazepines. Effects Lormetazepam (ATC N05CD06) has antianxiety, sedative, sleep-inducing, anticonvulsant, and muscle relaxant … Lormetazepam
Products Cinnarizine is commercially available in the form of capsules, tablets, and drops (Stugeron, generic). It has been approved in many countries since 1968. Since 2012, a fixed combination with dimenhydrinate has been on the market in many countries (Arlevert) see under Cinnarizine and Dimenhydrinate. Structure and properties Cinnarizine (C26H28N2, Mr = 368.51 g/mol) exists … Cinnarizine Effects and Side Effects
Products Flurazepam is commercially available in tablet form (Dalmadorm). It has been approved in many countries since 1972. Structure and properties Flurazepam (C21H23ClFN3O, Mr = 387.9 g/mol) is a 1,4-benzodiazepine. It is present in drugs as flurazepam hydrochloride, a white crystalline powder that is very soluble in water. Effects Flurazepam (ATC N05CD01) has sleep-inducing and … Flurazepam
Products Etomidate is commercially available as an emulsion for injection (etomidate lipuro). It has been approved in many countries since 1993. Structure and properties Etomidate (C14H16N2O2, Mr = 244.3 g/mol) is a pure -enantiomer. The imidazole-5-carboxylate ester is present as a white powder that is very sparingly soluble in water. Effects Etomidate (ATC N01AX07) has … Etomidate
Products Heroin (med. diamorphine) is commercially available as an injectable and in tablet form (Diaphin). It has been approved as a drug in many countries since 2001. Structure and properties Heroin is a diacetylated derivative of the opium ingredient morphine and belongs to the opioid group. It is present in drugs as diamorphine hydrochloride monohydrate … Heroin
Products Rupatadine is commercially available in tablet and oral solution forms (Rupafin, Urtimed), among others. The drug has not yet been registered in many countries. Structure and properties Rupatadine (C26H26ClN3, Mr = 415.96 g/mol) is present in drugs as rupatadine fumarate. It is structurally related to loratadine. Rupatadine is also partially metabolized to desloratadine but … Rupatadine
Products Flunitrazepam is commercially available in the form of film-coated tablets (Rohypnol). It has been approved in many countries since 1975. Structure and properties Flunitrazepam (C16H12FN3O3, Mr = 313.3 g/mol) is a lipophilic, fluorinated and nitrated 1,4-benzodiazepine. It exists as a white to yellowish crystalline powder that is practically insoluble in water. Effects Flunitrazepam (ATC … Flunitrazepam
Products Flupentixol is commercially available as film-coated tablets and as a solution for injection (Fluanxol). A fixed combination with melitracene is also available (Deanxit). The drug has been approved in many countries since 1967. See also under melitracene and flupentixol. Structure and properties Flupentixol (C23H25F3N2OS, Mr = 434.5 g/mol) is a thioxanthene derivative and a … Flupentixol
Products Amisulpride is commercially available as tablets, film-coated tablets, and a drinkable solution (Solian, generic). It has been approved in many countries since 1998. Structure and properties Amisulpride (C17H27N3O4S, Mr = 369.5 g/mol) is a substituted benzamide and a racemate. It exists as a white crystalline powder that is practically insoluble in water. Effects Amisulpride … Amisulpride
Products Tilidine is commercially available as an oral solution (Valoron). It has been approved in many countries since 1975. In Germany, tilidine fix is combined with the opioid antagonist naloxone to prevent abuse (Valoron N). Structure and properties Tilidine (C17H23NO2, Mr = 273.4 g/mol) is present in drugs as tilidine hydrochloride hemihydrate, a racemate and … Tilidine