Delorazepam

Products No medicines containing delorazepam are registered in many countries. In Italy, products available include EN drops and tablets and generics. Structure and properties Delorazepam (C15H10Cl2N2O, Mr = 305.2 g/mol) is a chlorinated and demethylated diazepam (Valium) related to lorazepam (Temesta). Effects Delorazepam (ATC N05BA) has antianxiety, sedative, anticonvulsant, and sleep-inducing properties. It crosses the … Delorazepam

Clenbuterol

Products Clenbuterol is not commercially available as a human drug in many countries, but exclusively as a veterinary drug for the treatment of respiratory diseases (e.g., Ventipulmin ad us vet). It is available only on medical prescription. In other countries, clenbuterol is on the market in tablet and drop form (Spiropent). Structure and properties Clenbuterol … Clenbuterol

Budesonide (Inhalation)

Products Budesonide is commercially available as a monopreparation for inhalation as a powder inhaler and suspension (Pulmicort, generics). It is also combined fixed with formoterol (Symbicort Turbuhaler, Vannair Dosage Aerosol). This article refers to monotherapy. Budesonide has been approved in many countries since 1988. Structure and properties Budesonide (C25H34O6, Mr = 430.5 g/mol) is a … Budesonide (Inhalation)

Budesonide Nasal Spray

Products Budesonide nasal sprays have been approved in many countries since 1995 (Cortinasal, generic). Rhinocort nasal spray has not been marketed since 2018. Sales of the Rhinocort turbuhaler were discontinued in 2020. Structure and properties Budesonide (C25H34O6, Mr = 430.5 g/mol) is a racemate and exists as a white, crystalline, odorless, tasteless powder that is … Budesonide Nasal Spray

Budesonide Capsules

Products Budesonide sustained-release capsules have been approved in many countries since 1998 (Entocort CIR, Budenofalk). Structure and properties Budesonide (C25H34O6, Mr = 430.5 g/mol) is a racemate and exists as a white, crystalline, odorless, tasteless powder that is practically insoluble in water. Effects Budesonide (ATC R03BA02) has anti-inflammatory, antiallergic, and immunosuppressive properties. The effects are … Budesonide Capsules

Citriodiol

Products Citriodiol is commercially available in the form of sprays (e.g. Anti-Brumm Naturel, Anti-Brumm Tick Stop + Icaridin), among others. Structure and properties Citriodiol is produced from an extract of leaves of lemon eucalyptus, also called (family: Myrtaceae). A major active ingredient is -menthane-3,8-diol (PMD, C10H20O2, Mr = 172.3 g/mol). Effects Citriodiol protects between 6-8 … Citriodiol

Bufexamac

Products Bufexamac was on the market in many countries as a cream and as an ointment (Parfenac). Because the active ingredient frequently causes allergic contact dermatitis, distribution of the drugs was discontinued. Structure and properties Bufexamac or 2-(4-butoxyphenyl)–hydroxyacetamide (C12H17NO3, Mr = 223.3 g/mol) is a white to almost white crystalline powder that is practically insoluble … Bufexamac

Citronella Oil

Products Citronella oil is commercially available in the form of sprays, bracelets, fragrance lamps and as pure essential oil, among other products. Structure and properties Citronella oil is the essential oil obtained by steam distillation from the fresh or partially dried aerial parts of (PhEur). It exists as a pale yellow to brownish yellow liquid … Citronella Oil

Buflomedil

Products Buflomedil is no longer available as a drug in many countries. Loftyl is out of commerce. Structure and properties Buflomedil (C17H25NO4, Mr = 307.4 g/mol) exists as a white, microcrystalline powder that is readily soluble in water. Effects Buflomedil (ATC C04AX20) is vasoactive and α-adrenolytic. It inhibits platelet aggregation, improves erythrocyte deformability and regional … Buflomedil

Citrulline

Products Citrulline is commercially available in the form of sachets containing a drinkable solution (Biostimol). It has been approved in many countries since 1996. Structure and properties L-(+)-citrulline (C6H13N3O3, Mr = 175.2 g/mol) exists as a white crystalline powder that is readily soluble in water. Citrulline is an amino acid found, for example, in watermelon. … Citrulline

Buformin

Products Buformin (Silubin retard, dragées) is no longer commercially available in many countries and many more because of the potential adverse effects. Structure and properties Buformin (C6H15N5, Mr = 157.2 g/mol) is a 1-butylbiguanide with a similar structure to metformin from the same drug group. It is present in drugs as buformin hydrochloride. Effects Buformin … Buformin

Cladribine

Products Cladribine was approved for the treatment of multiple sclerosis in the EU in 2017 and in the United States and many countries in 2019 in tablet form (Mavenclad). Cladribine has also been commercially available as an infusion and injection solution in many countries since 1998 (Litak). This article relates to MS therapy. Structure and … Cladribine